Properties
Description
ADL5859 HCl, soluble in DMSO, ethanol and water, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets δ-opioid receptor, κ-opioid receptor, and μ-opioid receptor.
Molecular Formula
C24H28N2O3·HCl
Targets
δ-Opioid receptor: 0.8 nM (Ki); κ-Opioid receptor: 37 nM (Ki); μ-Opioid receptor: 32 nM (Ki)
Solubility
DMSO: 76 mg/mL (177.17 mM); Water: 4 mg/mL (9.32 mM); Ethanol: 1 mg/mL (2.33 mM)
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
ADL5859 HCl can be used for its analgesic effects.
Storage
Store at -20℃, and keep desiccated.
