AhR inhibitor, Tapinarof, Purity ≥98%

Synonym: 79338-84-4; Benvitimod; WBI 1001; WBI1001; WBI-1001; GSK2894512; GSK 2894512; GSK-2894512; 5-[(E)-2-Phenylethenyl]-2-propan-2-ylbenzene-1,3-diol; AhR inhibitor

MDL: MFCD13193203
CAS Number: 79338-84-4
Compound CID: 6439522

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Tapinarof, soluble in DMSO and ethanol and insoluble in water, is an effective metabolism inhibitor, that has the ability to prevent the pathway of cell metabolism by inhibiting AhR. The molecular weight of the compound is 254.32, and its molecular formula is C₁₇H₁₈O₂.

Molecular Weight

254.32

Molecular Formula

C₁₇H₁₈O₂

Form

Lyophilized powder

Purity

≥98%

Impurities

Free from inappropriate visible particulates, foreign matter, discoloration, or other defects.

Solubility

In vitro: DMSO: 43 mg/mL (169.07 mM); Water: insoluble; Ethanol: 43 mg/mL (169.07 mM)

Identity

Confirmed by NMR/HPLC/MS.

Applications

Tapinarof can be used for its anti-inflammatory and immunomodulatory effects, making it a valuable therapeutic option in dermatology.