Properties
Description
Azasetron HCl, insoluble in DMSO and ethanol, and soluble in water, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets 5-HT3 receptor.
Molecular Formula
C17H20ClN3O3·HCl
Targets
5-HT3 receptor: 0.33 nM
Solubility
DMSO: insoluble; Water: 3 mg/mL (7.76 mM); Ethanol: insoluble
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
Azasetron HCl can be studied for its effect on blocking the action of serotonin, a neurotransmitter involved in triggering nausea and vomiting.
Storage
Store at -20°C, and keep desiccated.
