BQ-123

Synonym: 136553-81-6; Cyclo(D-trp-D-asp-pro-D-val-leu)

CAS Number: 136553-81-6
Compound CID: 443289

Product Size

2 mg; 5 mg; 10 mg; 20 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

BQ-123, soluble in DMSO and ethanol and insoluble in water, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets endothelin A receptor.

Molecular Weight

610.7

Molecular Formula

C₃₁H₄₂N₆O₇

Targets

Endothelin A receptor: 7.3 nM

Form

Lyophilized powder

Purity

>98%

Solubility

DMSO: 87 mg/mL (142.45 mM); Water: insoluble; Ethanol: 13 mg/mL (21.29 mM)

Applications

BQ-123 can be used for its ability to block endothelin receptors.