BTRX-335140

Synonym: 2244614-14-8; CYM-53093; Navacaprant

CAS Number: 2244614-14-8
Compound CID: 137434175

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

BTRX-335140 inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets δ opioid receptor/DOR, κ opioid receptor/KOR, and μ opioid receptor/MOR.

Molecular Weight

453.55

Molecular Formula

C₂₅H₃₂FN₅O₂

Targets

δ Opioid receptor/DOR: 6500 nM; κ Opioid receptor/KOR: 0.8 nM; μOpioid receptor/MOR: 110 nM

Form

Lyophilized powder

Purity

>98%

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

BTRX-335140 can be used for its antagonist activity for κOR, μOR and δOR.

Storage

Store at -20°C, and keep desiccated.