Properties
Description
BTRX-335140 inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets δ opioid receptor/DOR, κ opioid receptor/KOR, and μ opioid receptor/MOR.
Molecular Formula
C25H32FN5O2
Targets
δ Opioid receptor/DOR: 6500 nM; κ Opioid receptor/KOR: 0.8 nM; μOpioid receptor/MOR: 110 nM
Applications
BTRX-335140 can be used for its antagonist activity for κOR, μOR and δOR.