c-Ret inhibitor RET-IN-1, Purity ≥98%

Synonym: 2222755-14-6; RET-IN-1; SM0SJ89UOO; 4-(5-(6-((6-Methoxypyridin-3-yl)methyl)-3,6-diazabicyclo(3.1.1)heptan-3-yl)pyrazin-2-yl)-6-(((R)-morpholin-2-yl)methoxy)pyrazolo(1,5-a)pyridine-3-carbonitrile; c-Ret inhibitor

CAS Number: 2222755-14-6
Compound CID: 134437053

Product Size

1 mg; 2 mg; 5 mg; 10 mg; 25 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

RET-IN-1 primarily acts by blocking the ATP-binding site of the kinase domain of the RET protein, thereby inhibiting its autophosphorylation.

Molecular Weight

553.61

Molecular Formula

C₂₉H₃₁N₉O₃

Form

Lyophilized powder

Purity

≥98%

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

RET-IN-1 can be used to investigate the selective inhibition of RET kinase in cancer research.

Storage

Store at -20ºC.