Casein kinase inhibitor SR-3029, Purity ≥98%

Synonym: 1454585-06-8; Casein kinase inhibitor; SR 3029; SR3029

MDL: MFCD30187527
CAS Number: 1454585-06-8
Compound CID: 60196195

Product Size

2 mg; 5 mg; 10 mg; 25 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

SR-3029, soluble in DMSO and insoluble in ethanol and water, is a potent compound that inhibits Casein kinase activity. It targets CDK4/cyclin D1, CDK4/cyclin D3, CDK6/cyclin D1, CDK6/cyclin D3, CKIδ, and FLT3.

Molecular Weight

480.45

Molecular Formula

C₂₃H₁₉F₃N₈O

Targets

CDK4/cyclin D1: 576 nM; CDK4/cyclin D3: 368 nM; CDK6/cyclin D1: 428 nM; CDK6/cyclin D3: 427 nM; CKIδ: 44 nM; FLT3: 3000 nM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 43 mg/mL (89.49 mM); Water: Insoluble; Ethanol: Insoluble

Identity

Confirmed by NMR/HPLC/MS.

Applications

SR-3029 is a selective casein kinase 1δ/ε inhibitor, used in studying circadian rhythm regulation and potential cancer therapies.