CDK inhibitor Kenpaullone, Purity ≥98%

Synonym: 142273-20-9; Kenpaullone; 9-Bromopaullone; NSC 664704; NSC-664704; CDK inhibitor

CAS Number: 142273-20-9
Compound CID: 3820

Product Size

10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Kenpaullone, soluble in DMSO and insoluble in ethanol and water, is an CDK kinase inhibitor that disrupts cell division processes. It targets CDK1/CyclinB, CDK2/CyclinA, c-Src, and CaseinKinase2.

Molecular Weight

327.2

Molecular Formula

C₁₆H₁₁BrN₂O

Targets

CDK1/CyclinB: 0.4 μM; CDK2/CyclinA: 0.68 μM; c-Src: 15 μM; CaseinKinase2: 20 μM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 58 mg/mL (177.27 mM; Water: Insoluble; Ethanol: Insoluble

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

Kenpaullone can be used to investigate its role as a CDK inhibitor and its potential effects on cell cycle regulation and apoptosis.

Storage

Store at -20ºC.