CDK inhibitor LY2857785, Purity ≥98%

Synonym: 1619903-54-6; LY-2857785; LY 2857785; CDK inhibitor

CAS Number: 1619903-54-6
Compound CID: 78357764

Product Size

5 mg; 10 mg; 25 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

LY2857785, soluble in DMSO and ethanol and insoluble in water, is an CDK kinase inhibitor that disrupts cell division processes. It targets CDK7, CDK8, and CDK9.

Molecular Weight

448.6

Molecular Formula

C₂₆H₃₆N₆O

Targets

CDK7: 0.246 μM; CDK8: 0.016 μM; CDK9: 0.011 μM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 22 mg/mL (49.04 mM); Water: Insoluble; Ethanol: 40 mg/mL (89.16 mM)

Identity

Confirmed by NMR/HPLC/MS.

Applications

LY2857785 can be utilized in research on the inhibition of CDKs with implications for cancer therapy.