Properties
Description
CGS-15943 inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets adenosine A1 receptor, adenosine A2A receptor, adenosine A2B receptor, adenosine A3 receptor, p110δ, and p110γ.
Molecular Formula
C13H8ClN5O
Targets
Adenosine A1 receptor: 3.5 nM; Adenosine A2A receptor: 4.2 nM; Adenosine A2B receptor: 16 nM; Adenosine A3 receptor: 50 nM; p110δ: 8.47 μM; p110γ: 1.1 μM
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
CGS-15943 can be used for research on the role of adenosine receptors in various physiological and pathological processes in the central nervous system.
Storage
Store at -20°C, and keep desiccated.
