Properties
Description
CP 945598 HCl (otenabant HCl), soluble in DMSO and insoluble in water and ethanol, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets hCB1, hCB2, and rCB1.
Molecular Formula
C25H25Cl2N7O·HCl
Targets
hCB1: 0.7 nM (Ki); hCB2: 7.663 μM (Ki); rCB1: 2.8 nM (Ki)
Solubility
DMSO: 5 mg/mL (9.14 mM); Water: insoluble; Ethanol: insoluble
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
CP 945598 HCl (otenabant HCl) can be used for its anti-inflammatory and immunomodulatory effects.
Storage
Store at -20°C, and keep desiccated.
