Properties
Description
Derenofylline inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets A1R, A2AR, and adenosine A3 receptor.
Molecular Formula
C18H20N4O
Targets
A1R: 1 nM; A2AR: 398 nM; Adenosine A3 receptor: 200 nM
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
Derenofylline can be used for its ability to antagonize CRF-stimulated adenylate cyclase activity.
Storage
Store at -20°C, and keep desiccated.
