DGAT inhibitor, PF-04620110, Purity ≥98%

Synonym: 1109276-89-2; PF04620110; PF 04620110; 2-[4-[4-(4-Amino-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6-yl)phenyl]cyclohexyl]acetic acid; DGAT inhibitor

CAS Number: 1109276-89-2
Compound CID: 46926360

Product Size

10 mg; 25 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

PF-04620110, soluble in DMSO and insoluble in water and ethanol, is an effective metabolism inhibitor, that has the ability to prevent the pathway of cell metabolism by inhibiting DGAT. The molecular weight of the compound is 396.44, and its molecular formula is C₂₁H₂₄N₄O₄. It targets the DGAT1.

Molecular Weight

396.44

Molecular Formula

C₂₁H₂₄N₄O₄

Targets

DGAT1

Form

Lyophilized powder

Purity

≥98%

Impurities

Free from inappropriate visible particulates, foreign matter, discoloration, or other defects.

Solubility

In vitro: DMSO (warmed): 46 mg/mL (116.03 mM); Water: insoluble; Ethanol: insoluble

Identity

Confirmed by NMR/HPLC/MS.

Applications

PF-04620110 can be studied extensively for its potential therapeutic applications in the treatment of various cancers, particularly those with dysregulated PI3K/mTOR signaling pathways。