E3 ligase ligand-linker conjugate inhibitor, (S,R,S)-AHPC-PEG4-NH₂, Purity ≥98%

Synonym: 2010159-57-4; VH032-PEG4-NH₂; VHL ligand-linker conjugate 4; E3 ligase ligand-linker conjugate 7 free base; (2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-(2-Aminoethoxy)ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; E3 ligase ligand-linker conjugate inhibitor

CAS Number: 2010159-57-4
Compound CID: 124177628

Product Size

100 mg; 200 mg; 500 mg; 1 g

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

(S,R,S)-AHPC-PEG4-NH₂ is an effective PROTAC inhibitor, that has the ability to prevent the pathway of E3 ligase ligand-linker conjugation. The molecular weight of the compound is 663.83, and its molecular formula is C₃₂H₄₉N₅O₈S.

Molecular Weight

663.83

Molecular Formula

C₃₂H₄₉N₅O₈S

Form

Lyophilized powder

Purity

≥98%

Impurities

Free from inappropriate visible particulates, foreign matter, discoloration, or other defects.

Identity

Confirmed by NMR/HPLC/MS.

Applications

(S,R,S)-AHPC-PEG4-NH₂ plays a key role in enhancing the pharmacological properties of linked drugs.

E3 ligase ligand-linker conjugate inhibitor, (S,R,S)-AHPC-PEG4-NH2, Purity ≥98%

E3 ligase ligand-linker conjugate inhibitor, (S,R,S)-AHPC-PEG4-NH₂, Purity ≥98%