Eletriptan hydrobromide

Synonym: 177834-92-3; Eletriptan HBr; Relpax

CAS Number: 177834-92-3
Compound CID: 656631

Product Size

10 mg; 25 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Eletriptan hydrobromide, soluble in DMSO and insoluble in water and ethanol, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets 5-HT1B, and 5-HT1D.

Molecular Weight

463.43

Molecular Formula

C₂₂H₂₆N₂O₂S·HBr

Targets

5-HT1B: 0.92 nM (Ki); 5-HT1D: 3.14 nM (Ki)

Form

Lyophilized powder

Purity

>98%

Solubility

DMSO: 83 mg/mL (179.09 mM); Water: insoluble; Ethanol: insoluble

Applications

Eletriptan hydrobromide can be used to research and develop therapeutic strategies for certain diseases that involve excessive activation of GPCR-G protein signaling pathways.