Epigenetic reader domain inhibitor Alobresib, Purity ≥98%

Synonym: 1637771-14-2; GS-5829; GS 5829; GS5829; Epigenetic reader domain inhibitor

CAS Number: 1637771-14-2
Compound CID: 86281210

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Alobresib, soluble in DMSO, water and ethanol, disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals.

Molecular Weight

437.49

Molecular Formula

C₂₆H₂₃N₅O₂

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 76 mg/mL (173.72 mM); Water: <1 mg/mL; Ethanol: 10 mg/mL (22.85 mM)

Identity

Confirmed by NMR/HPLC/MS.

Applications

Alobresib can be used to investigate the inhibition of BET bromodomains, studying their potential as cancer therapeutics through modulation of gene expression.