Properties
Description
Apabetalone, soluble in DMSO and insoluble in ethanol and water, disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals. It targets BD2.
Molecular Formula
C20H22N2O5
Solubility
DMSO: 63 mg/mL (170.08 mM); Water: Insoluble; Ethanol: Insoluble
Identity
Confirmed by NMR/HPLC/MS.
Applications
Apabetalone can be used to investigate the inhibition of BET bromodomains, focusing on therapeutic potential in cardiovascular and metabolic diseases.