Epigenetic reader domain inhibitor BET-IN-1, Purity ≥98%

Synonym: 1422554-34-4; BET-IN-1; I-BET282; CHEMBL4878439; (R)-4-(8-methoxy-1-(1-methoxypropan-2-yl)-2-(tetrahydro-2H-pyran-4-yl)-1H-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole; Epigenetic reader domain inhibitor

CAS Number: 1422554-34-4
Compound CID: 71258968

Product Size

1 mg; 5 mg; 10 mg; 50 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

BET-IN-1 disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals.

Molecular Weight

450.53

Molecular Formula

C₂₅H₃₀N₄O₄

Form

Lyophilized powder

Purity

≥98%

Identity

Confirmed by NMR/HPLC/MS.

Applications

BET-IN-1 can be used to investigate the inhibition of BET bromodomains and the consequent effects on gene transcriptional activity.