Properties
Description
BI-9564, soluble in DMSO and ethanol and insoluble in water, disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals. It targets BRD7, BRD9, and CECR2.
Molecular Formula
C20H23N3O3
Targets
BRD7: 73 nM (Kd); BRD9: 5.9 nM (Kd); CECR2: 77 nM (Kd)
Solubility
DMSO: 3 mg/mL (8.48 mM); Water: Insoluble; Ethanol: 15 mg/mL (42.44 mM)
Identity
Confirmed by NMR/HPLC/MS.
Applications
BI-9564 can be used to study the inhibition of specific bromodomains, contributing to research on gene regulation and disease.
