Epigenetic reader domain inhibitor BI-9564, Purity ≥98%

Synonym: 1883429-22-8; BI 9564; BI9564; Epigenetic reader domain inhibitor

CAS Number: 1883429-22-8
Compound CID: 117072549

Product Size

5 mg; 10 mg; 50 mg

Price

Datasheet

MSDS

Properties

Description

BI-9564, soluble in DMSO and ethanol and insoluble in water, disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals. It targets BRD7, BRD9, and CECR2.

Molecular Weight

353.41

Molecular Formula

C₂₀H₂₃N₃O₃

Targets

BRD7: 73 nM (Kd); BRD9: 5.9 nM (Kd); CECR2: 77 nM (Kd)

Form

Lyophilized powder

Purity

Solubility

DMSO: 3 mg/mL (8.48 mM); Water: Insoluble; Ethanol: 15 mg/mL (42.44 mM)

Identity

Confirmed by NMR/HPLC/MS.

Applications

BI-9564 can be used to study the inhibition of specific bromodomains, contributing to research on gene regulation and disease.