Epigenetic reader domain inhibitor CPI 0610, Purity ≥98%

Synonym: 1380087-89-7; CPI0610; CPI-0610; Epigenetic reader domain inhibitor

CAS Number: 1380087-89-7
Compound CID: 57389999

Product Size

5 mg; 10 mg; 50 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

CPI 0610, soluble in DMSO and ethanol and insoluble in water, disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals. It targets BRD4-BD1, and MYC.

Molecular Weight

365.82

Molecular Formula

C₂₀H₁₆ClN₃O₂

Targets

BRD4-BD1: 39 nM; MYC: 180 nM (EC₅₀)

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 70 mg/mL (191.35 mM); Water: Insoluble; Ethanol: 12 mg/mL

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

CPI 0610 can be used to study the therapeutic potential of BET inhibition in hematologic malignancies.

Storage

Store at -20ºC.