Properties
Description
CPI-637, soluble in DMSO and insoluble in ethanol and water, disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals. It targets BRD4 BD1.
Molecular Formula
C22H22N6O
Solubility
DMSO: 27 mg/mL (69.86 mM); Water: Insoluble; Ethanol: Insoluble
Identity
Confirmed by NMR/HPLC/MS.
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
CPI-637 can be used to study the effects of BET inhibition on gene expression and oncogenesis.