Epigenetic reader domain inhibitor GNE-207, Purity ≥98%

Synonym: 2158266-58-9; GNE207; GNE 207; Epigenetic reader domain inhibitor

CAS Number: 2158266-58-9
Compound CID: 132186469

Product Size

1 mg; 5 mg; 10 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

GNE-207 disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals. It targets BRD4 (1) and CBP.

Molecular Weight

510.6

Molecular Formula

C₂₉H₃₀N₆O₃

Targets

BRD4 (1): 3.1 μM; CBP: 1 μM

Form

Lyophilized powder

Purity

≥98%

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

GNE-207 can be used to study the inhibition of bromodomains in the context of gene regulation and disease.

Storage

Store at -20ºC.