Properties
Description
GSK 5959, soluble in DMSO and ethanol and insoluble in water, disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals.
Molecular Formula
C22H26N4O3
Solubility
DMSO: 5 mg/mL (12.68 mM); Water: Insoluble; Ethanol: 3 mg/mL (7.6 mM)
Identity
Confirmed by NMR/HPLC/MS.
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
GSK 5959 can be used to investigate the role of BET bromodomains in gene expression and cancer.
