Properties
Description
GSK6853, soluble in warmed DMSO and warmed ethanol and insoluble in water, disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals.
Molecular Formula
C22H27N5O3
Solubility
Warmed DMSO: 77 mg/mL (188.04 mM); Water: Insoluble; Warmed ethanol: 77 mg/mL (188.04 mM)
Identity
Confirmed by NMR/HPLC/MS.
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
GSK6853 can be used to explore the impact of BET bromodomain inhibition on gene expression and disease.