Properties
Description
TP-472 disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals. It targets BRD7 and BRD9.
Molecular Formula
C20H19N3O2
Targets
BRD7: 0.34 μM (Kd); BRD9: 33 μM (Kd)
Identity
Confirmed by NMR/HPLC/MS.
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
TP-472 is employed to explore the role of BET bromodomain inhibition in disease contexts.