Eplivanserin

Synonym: 130579-75-8; SR-46349; SR 46349; SR46349

CAS Number: 130579-75-8
Compound CID: 135456190

Product Size

1 mg; 5 mg; 10 mg; 50 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Eplivanserin inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets 5-HT2A receptor, 5-HT2A receptor, and 5-HT2C receptor.

Molecular Weight

328.38

Molecular Formula

C₁₉H₂₁FN₂O₂

Targets

5-HT2A receptor: 5.8 nM (IC₅₀, in rat cortical membrane); 5-HT2A receptor: 1.14 nM; 5-HT2C receptor: 120 nM

Form

Lyophilized powder

Purity

>98%

Applications

Eplivanserin can be used for its ability to promote sleep induction and improve sleep quality in patients with insomnia.