Properties
Description
Eplivanserin inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets 5-HT2A receptor, 5-HT2A receptor, and 5-HT2C receptor.
Molecular Formula
C19H21FN2O2
Targets
5-HT2A receptor: 5.8 nM (IC50, in rat cortical membrane); 5-HT2A receptor: 1.14 nM; 5-HT2C receptor: 120 nM
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
Eplivanserin can be used for its ability to promote sleep induction and improve sleep quality in patients with insomnia.
Storage
Store at -20°C, and keep desiccated.
