ERK inhibitor DEL-22379, Purity ≥98%

Synonym: DEL-22379; 181223-80-3; CHEMBL5180742; (Z)-N-(3-((5-Methoxy-1H-indol-3-yl)methylene)-2-oxoindolin-5-yl)-3-(piperidin-1-yl)propanamide; N-[(3Z)-3-[(5-Methoxy-1H-indol-3-yl)methylidene]-2-oxo-1H-indol-5-yl]-3-piperidin-1-ylpropanamide; ERK inhibitor

CAS Number: 181223-80-3
Compound CID: 11224574

Product Size

5 mg; 10 mg; 25 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

DEL-22379, soluble in DMSO and insoluble in ethanol and water, exhibits potent inhibition of ERK kinase. It targets ERK.

Molecular Weight

444.55

Molecular Formula

C₂₆H₂₈N₄O₃

Targets

ERK: 0.5 μM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 79 mg/mL (177.71 mM); Water: Insoluble; Ethanol: Insoluble

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

DEL-22379 can be used to explore the inhibition of ERK dimerization and its effects on cellular functions.

Storage

Store at -20ºC.