Factor Xa inhibitor, Tosylate monohydrate, Purity ≥98%

Synonym: 1229194-11-9; DU-176b; Edoxaban tosylate hydrate; Edoxaban tosylate monohydrate; Lixiana; N'-(5-Chloropyridin-2-yl)-N-[(1S,2R,4S)-4-(dimethylcarbamoyl)-2-[(5-methyl-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-2-carbonyl)amino]cyclohexyl]oxamide; 4-methylbenzenesulfonic acid; hydrate; Factor Xa inhibitor

MDL: MFCD28400751
CAS Number: 1229194-11-9
Compound CID: 25022378

Product Size

10 mg; 25 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Tosylate monohydrate, soluble in DMSO and insoluble in water and ethanol, is an effective metabolism inhibitor, that has the ability to prevent the pathway of cell metabolism by inhibiting factor Xa. The molecular weight of the compound is 738.27, and its molecular formula is C₂₄H₃₀ClN₇O₄S·C₇H₈O₃S·H₂O. It targets the Factor Xa, FIXa and Thrombin.

Molecular Weight

738.27

Molecular Formula

C₂₄H₃₀ClN₇O₄S·C₇H₈O₃S·H₂O

Targets

Factor Xa

Form

Lyophilized powder

Purity

≥98%

Impurities

Free from inappropriate visible particulates, foreign matter, discoloration, or other defects.

Solubility

In vitro: DMSO: 89 mg/mL (120.55 mM); Water: insoluble; Ethanol: insoluble

Identity

Confirmed by NMR/HPLC/MS.

Applications

Tosylate monohydrate displays the significant potential to act as an effective bioavailable pyrazole antithrombotic agent.