FGFR inhibitor E-3810, Purity ≥98%

Synonym: 1058137-23-7; FGFR inhibitor; E 3810; E3810; Lucitanib

CAS Number: 1058137-23-7
Compound CID: 25031915

Product Size

5 mg; 10 mg; 50 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

E-3810 is a protein tyrosine kinase inhibitor that has shown potent biochemical activity against FGFR. It targets FGFR1, FGFR2, VEGFR1, VEGFR2, and VEGFR3.

Molecular Weight

443.49

Molecular Formula

C₂₆H₂₅N₃O₄

Targets

FGFR1: 17.5 nM; FGFR2: 82.5 nM; VEGFR1: 7 nM; VEGFR2: 25 nM; VEGFR3: 10 nM

Form

Lyophilized powder

Purity

≥98%

Identity

Confirmed by NMR/HPLC/MS.

Applications

E-3810 serves as a research compound to inhibit FGFR, helping to deepen insights into FGFR-associated cancers and potential therapeutic interventions.