Glucokinase inhibitor, LY2608204, Purity ≥98%

Synonym: 1234703-40-2; LY-2608204; (1R,2S)-2-Cyclohexyl-1-(4-cyclopropylsulfonylphenyl)-N-[5-(2-pyrrolidin-1-ylethylsulfanyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide; Glucokinase inhibitor

MDL: MFCD21609257
CAS Number: 1234703-40-2
Compound CID: 46832368

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

MSDS

Properties

Description

LY2608204, soluble in DMSO and ethanol and insoluble in water, is a glucose kinase (GK) activator. The molecular weight of the compound is 559.8, and its molecular formula is C₂₈H₃₇N₃O₃S₃. It targets the glucokinase.

Molecular Weight

559.8

Molecular Formula

C₂₈H₃₇N₃O₃S₃

Targets

Glucokinase

Form

Lyophilized powder

Purity

Impurities

Free from inappropriate visible particulates, foreign matter, discoloration, or other defects.

Solubility

In vitro: DMSO: 95 mg/mL (169.69 mM); Water: insoluble; Ethanol: 30 mg/mL (53.59 mM); In vivo: 1% DMSO + 30% polyethylene glycol + 1% Tween 80, 28 mg/mL

Identity

Confirmed by NMR/HPLC/MS.

Applications

LY2608204 plays a key role in disrupting the signaling pathways that promote tumor growth.