GnRH receptor inhibitor Relugolix, Purity ≥98%

Synonym: 737789-87-6; GnRH receptor inhibitor; TAK385; TAK-385; TAK 385; Relugolix

MDL: MFCD25976856
CAS Number: 737789-87-6
Compound CID: 10348973

Product Size

1 mg; 5 mg; 10 mg; 50 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Relugolix, soluble in DMSO and insoluble in ethanol and water, is a compound that blocks the GnRH receptor, a G-protein coupled receptor involved in the regulation of reproductive hormone release from the pituitary gland, with implications for the treatment of conditions like hormone-sensitive cancers and infertility.

Molecular Weight

623.63

Molecular Formula

C₂₉H₂₇F₂N₇O₅S

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 59 mg/mL (94.6 mM); Water: Insoluble; Ethanol: Insoluble

Identity

Confirmed by NMR/HPLC/MS.

Applications

Relugolix is used for research on GnRH pathways, with applications in treating hormone-sensitive conditions.