GSK163090

Synonym: 844903-58-8; 1-(3-(2-(4-(2-Methyl-5-quinolinyl)-1-piperazinyl)ethyl)phenyl)-2-imidazolidinone

CAS Number: 844903-58-8
Compound CID: 11292933

Product Size

5 mg; 10 mg; 25 mg; 50 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

GSK163090 inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets 5-HT1A receptor, 5-HT1B receptor, 5-HT1D receptor, 5-HT2A receptor, 5-HT2B receptor, 5-HT2C receptor, D2 receptor, D3 receptor, human 5-HT6 receptor, and human 5-HT7 receptor.

Molecular Weight

415.53

Molecular Formula

C₂₅H₂₉N₅O

Targets

5-HT1A receptor: 9.4 (pKi); 5-HT1B receptor: 8.5 (pKi); 5-HT1D receptor: 9.7 (pKi); 5-HT2A receptor: 6 (pKi); 5-HT2B receptor: 6.3 (pKi); 5-HT2C receptor: 5.8 (pKi); D2 receptor: 6.3 (pKi); D3 receptor: 6.7 (pKi); Human 5-HT6 receptor: <5.3 (pKi); Human 5-HT7 receptor: 6.8 (pKi)

Form

Lyophilized powder

Purity

>98%

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

GSK163090 can be used for its effects on neurological function and its potential role in modulating neurotransmitter systems within the brain.

Storage

Store at -20°C, and keep desiccated.