GSK163090

Synonym: 844903-58-8; 1-(3-(2-(4-(2-Methyl-5-quinolinyl)-1-piperazinyl)ethyl)phenyl)-2-imidazolidinone

CAS Number: 844903-58-8
Compound CID: 11292933

Product Size

5 mg; 10 mg; 25 mg; 50 mg

Price

Datasheet

MSDS

Properties

Description

GSK163090 inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets 5-HT1A receptor, 5-HT1B receptor, 5-HT1D receptor, 5-HT2A receptor, 5-HT2B receptor, 5-HT2C receptor, D2 receptor, D3 receptor, human 5-HT6 receptor, and human 5-HT7 receptor.

Molecular Weight

415.53

Molecular Formula

C₂₅H₂₉N₅O

Targets

5-HT1A receptor: 9.4 (pKi); 5-HT1B receptor: 8.5 (pKi); 5-HT1D receptor: 9.7 (pKi); 5-HT2A receptor: 6 (pKi); 5-HT2B receptor: 6.3 (pKi); 5-HT2C receptor: 5.8 (pKi); D2 receptor: 6.3 (pKi); D3 receptor: 6.7 (pKi); Human 5-HT6 receptor: <5.3 (pKi); Human 5-HT7 receptor: 6.8 (pKi)

Form

Lyophilized powder

Purity

Applications

GSK163090 can be used for its effects on neurological function and its potential role in modulating neurotransmitter systems within the brain.