Properties
Description
H4R antagonist 1 inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets human H4 receptor, and mouse H4 receptor.
Molecular Formula
C11H11BrN8
Targets
Human H4 receptor: 27 nM; Mouse H4 receptor: 290 nM
Applications
H4R antagonist 1 can be used for its anti-itching and anti-inflammation activity.