Properties
Description
BIX 01294, soluble in DMSO, water and ethanol, inhibits the enzymes that add methyl groups to histone proteins, altering chromatin structure and gene expression.
Molecular Formula
C28H38N6O2.3HCl
Solubility
DMSO: 95 mg/mL (158.32 mM); Water: 95 mg/mL (158.32 mM); Ethanol: 8 mg/mL
Identity
Confirmed by NMR/HPLC/MS.
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
BIX 01294 can be used to inhibit G9a histone methyltransferase, which is involved in epigenetic regulation.
