HMT inhibitor PFI-2, Purity ≥98%

Synonym: 1627676-59-8; PFI2; Histone methyltransferase inhibitor

Product Size

10 mg; 25 mg; 50 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

PFI-2 inhibits the enzymes that add methyl groups to histone proteins, altering chromatin structure and gene expression. It targets SETD7 and SETD7.

Molecular Weight

499.52

Molecular Formula

C₂₃H₂₅F₄N₃O₃S

Targets

SETD7: 0.33 nM (Ki); SETD7: 2 nM

Form

Lyophilized powder

Purity

≥98%

Identity

Confirmed by NMR/HPLC/MS.

Applications

PFI-2 can be used to inhibit the SETD7 methyltransferase, studying its role in cellular processes and disease.