Properties
Description
WDR5-0103, soluble in DMSO and ethanol and insoluble in water, inhibits the enzymes that add methyl groups to histone proteins, altering chromatin structure and gene expression.
Molecular Formula
C21H25N3O4
Solubility
DMSO: 68 mg/mL (177.34 mM); Water: Insoluble; Ethanol: 18 mg/mL (46.94 mM)
Identity
Confirmed by NMR/HPLC/MS.
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
WDR5-0103 can be used to disrupt the interaction of WDR5 with histone-modifying complexes, affecting gene regulation.
