Hydroxylase inhibitor, Enarodustat, Purity ≥98%

Synonym: 1262132-81-9; JTZ-951; JTZ 951; JTZ951; 2-[[7-Oxo-5-(2-phenylethyl)-3H-[1,2,4]triazolo[1,5-a]pyridine-8-carbonyl]amino]acetic acid; Hydroxylase inhibitor

CAS Number: 1262132-81-9
Compound CID: 50899324

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Enarodustat, soluble in DMSO and ethanol and insoluble in water, is an effective metabolism inhibitor, that has the ability to prevent the pathway of cell metabolism by inhibiting hydroxylases. The molecular weight of the compound is 340.33, and its molecular formula is C₁₇H₁₆N₄O₄.

Molecular Weight

340.33

Molecular Formula

C₁₇H₁₆N₄O₄

Form

Lyophilized powder

Purity

≥98%

Impurities

Free from inappropriate visible particulates, foreign matter, discoloration, or other defects.

Solubility

In vitro: DMSO: 67 mg/mL (196.86 mM); Water: insoluble; Ethanol: 2 mg/mL (5.87 mM)

Identity

Confirmed by NMR/HPLC/MS.

Applications

Enarodustat can be studied extensively for its potential therapeutic applications in the treatment of anemia, particularly in chronic kidney disease, by stimulating erythropoiesis and improving hemoglobin levels.