Isocitrate dehydrogenase (IDH) inhibitor, GSK864, Purity ≥98%

Synonym: 1816331-66-4; GSK 864; GSK-864; (7S)-1-[(4-Fluorophenyl)methyl]-3-N-(4-methoxy-3,5-dimethylphenyl)-7-methyl-5-(1H-pyrrole-2-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3,7-dicarboxamide; Isocitrate dehydrogenase (IDH) inhibitor

CAS Number: 1816331-66-4
Compound CID: 91864701

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

GSK864 is an effective metabolism inhibitor, that has the ability to prevent the pathway of cell metabolism by inhibiting isocitrate dehydrogenase (IDH). The molecular weight of the compound is 558.6, and its molecular formula is C₃₀H₃₁FN₆O₄.

Molecular Weight

558.6

Molecular Formula

C₃₀H₃₁FN₆O₄

Form

Lyophilized powder

Purity

≥98%

Impurities

Free from inappropriate visible particulates, foreign matter, discoloration, or other defects.

Identity

Confirmed by NMR/HPLC/MS.

Applications

GSK864 plays a key role in inhibiting the mutant IDH1 enzyme, which is involved in cancer progression.