Ki16198

Synonym: 355025-13-7; Methyl 3-((4-(4-(((1-(2-chlorophenyl)ethoxy)carbonyl)amino)-3-methylisoxazol-5-yl)benzyl)thio)propanoate

CAS Number: 355025-13-7
Compound CID: 9913405

Product Size

5 mg; 10 mg; 25 mg; 50 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Ki16198, soluble in DMSO and ethanol and insoluble in water, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets LPA1, and LPA3.

Molecular Weight

488.98

Molecular Formula

C₂₄H₂₅ClN₂O₅S

Targets

LPA1: 0.34 μM (Ki); LPA3: 0.93 μM (Ki)

Form

Lyophilized powder

Purity

>98%

Solubility

DMSO: 86 mg/mL (175.87 mM); Water: insoluble; Ethanol: 32 mg/mL (65.44 mM)

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

Ki16198 can be used as a selective antagonist of the serotonin 5-HT6 receptor.

Storage

Store at -20°C, and keep desiccated.