Properties
Description
MK-1064, soluble in DMSO and insoluble in water and ethanol, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets OX1 receptor, OX1 receptor, OX2 receptor, and OX2 receptor.
Molecular Formula
C24H20ClN5O3
Targets
OX1 receptor: 1789 nM; OX1 receptor: 1584 nM; OX2 receptor: 18 nM; OX2 receptor: 0.5 nM
Solubility
DMSO: 87 mg/mL (188.35 mM); Water: insoluble; Ethanol: insoluble
Stability
The product is stable for three years when stored at the recommended temperature in lyophilized powder.
Applications
MK-1064 can be used for its anti-cancer properties.
Storage
Store at -20°C, and keep desiccated.