MK-1064

Synonym: 1207253-08-4; 5''-Chloro-N-[(5,6-dimethoxypyridin-2-yl)methyl]-2,2':5',3''-terpyridine-3'-carboxamide

CAS Number: 1207253-08-4
Compound CID: 44633765

Product Size

1 mg; 2 mg; 5 mg; 10 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

MK-1064, soluble in DMSO and insoluble in water and ethanol, inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets OX1 receptor, OX1 receptor, OX2 receptor, and OX2 receptor.

Molecular Weight

461.91

Molecular Formula

C₂₄H₂₀ClN₅O₃

Targets

OX1 receptor: 1789 nM; OX1 receptor: 1584 nM; OX2 receptor: 18 nM; OX2 receptor: 0.5 nM

Form

Lyophilized powder

Purity

>98%

Solubility

DMSO: 87 mg/mL (188.35 mM); Water: insoluble; Ethanol: insoluble

Applications

MK-1064 can be used for its anti-cancer properties.