p53 inhibitor APR-246, Purity ≥98%

Synonym: 5291-32-7; APR-246; PRIMA-1MET; Eprenetapopt; 2-(Hydroxymethyl)-2-(methoxymethyl)-1-azabicyclo[2.2.2]octan-3-one; 2-(Hydroxymethyl)-2-(methoxymethyl)quinuclidin-3-one; p53 inhibitor

MDL: MFCD16294187; MFCD20620963
CAS Number: 5291-32-7
Compound CID: 52918385

Product Size

10 mg; 25 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

APR-246, soluble in DMSO, water and ethanol, is a compound with potential antineoplastic activity.

Molecular Weight

199.24688

Molecular Formula

C₁₀H₁₇NO₃

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 38 mg/mL (190.71 mM); Water: 38 mg/mL (190.71 mM); Ethanol: 38 mg/mL

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

APR-246 can be used to restore the function of mutant p53, aiding in the development of targeted cancer therapies.

Storage

Store at -20ºC.