PAD inhibitor GSK199, Purity ≥98%

Synonym: 1549811-53-1; GSK199; (R)-(3-Aminopiperidin-1-yl)(2-(1-ethyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-7-methoxy-1-methyl-1H-benzo[d]imidazol-5-yl)methanone hydrochloride; GSK-199; GSK199 hydrochloride; Protein arginine deiminase (PAD) inhibitor

CAS Number: 1549811-53-1
Compound CID: 86340155

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

GSK199 prevents the conversion of arginine residues to citrulline in proteins, which is important in processes like gene regulation and inflammatory responses.

Molecular Weight

468.98

Molecular Formula

C₂₄H₂₉ClN₆O₂

Form

Lyophilized powder

Purity

≥98%

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

GSK199 can be used to study activity of histone methyltransferase EZH2 in cancer therapy trials.

Storage

Store at -20ºC.