PAK inhibitor, LOR-253, Purity ≥98%

Cat. No.: X24-08-YM271

PAK inhibitor, LOR-253, Purity ≥98%

Synonym: 916151-99-0; LOR 253; LOR253; APTO-253; 2-(5-Fluoro-2-methyl-1H-indol-3-yl)-1H-imidazo[4,5-f][1,10]phenanthroline

  • CAS Number: 916151-99-0
  • Compound CID: 11960271
Product Size
10 mg; 25 mg; 50 mg; 100 mg
Price
Datasheet
MSDS
Properties
Description
LOR-253, soluble in DMSO and insoluble in water and ethanol, is an effective cytoskeleton inhibitor, that has the ability to prevent the pathway of cytoskeletal signaling by inhibiting PAK.
Molecular Weight
367.38
Molecular Formula
C22H14FN5
Form
Lyophilized powder
Purity
≥98%
Titer
Free from inappropriate visible particulates, foreign matter, discoloration, or other defects
Solubility
In vitro: DMSO: 72 mg/mL (195.98 mM); Water: insoluble; Ethanol: insoluble
Stability
In its lyophilized form, the chemical remains stable for 36 months.
Quality Level
Research grade
Applications
LOR-253 is a cytoskeletal signaling inhibitor that can be studied extensively for its potential therapeutic applications in the treatment of various cancers and fibrotic diseases by blocking TGF-β signaling, which plays a role in tumor progression and fibrosis.
Storage
Store at -20ºC, and keep desiccated.
Related Products

About Us

CD BioGlyco is a world-class biotechnology company with offices in many countries. Our products and services provide a viable option to what is otherwise available.

Contact Us

Copyright © CD BioGlyco. All rights reserved.