PARP inhibitor GeA-69, Purity ≥98%

Synonym: 2143475-98-1; GeA-69; N-(2-(9H-Carbazol-1-yl)phenyl)acetamide;N-[2-(9H-Carbazol-1-yl)phenyl]acetamide; PARP inhibitor

CAS Number: 2143475-98-1
Compound CID: 135397654

Product Size

5 mg; 10 mg; 25 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

GeA-69, soluble in DMSO and ethanol and insoluble in water, binds to the PARP enzyme's active site, preventing it from repairing single-strand DNA breaks.

Molecular Weight

300.35

Molecular Formula

C₂₀H₁₆N₂O

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 52 mg/mL (173.13 mM); Water: Insoluble; Ethanol: 9 mg/mL (29.96 mM)

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

GeA-69 can be used to explore its role as an inhibitor of tankyrase, impacting Wnt/β-catenin signaling.

Storage

Store at -20ºC.