PDGFR inhibitor CP-868596, Purity ≥98%

Synonym: 670220-88-9; PDGFR inhibitor; CP868596; CP 868596

MDL: MFCD21609260
CAS Number: 670220-88-9
Compound CID: 10366136

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

CP-868596, soluble in warmed DMSO and ethanol and insoluble in water, blocks the activity of platelet-derived growth factor receptors (PDGFR), which play a crucial role in cell growth, angiogenesis, and tissue. It targets FLT3, PDGFRα (CHO cells), and PDGFRβ (CHO cells).

Molecular Weight

443.5

Molecular Formula

C₂₆H₂₉N₅O₂

Targets

FLT3: 0.74 nM (Kd); PDGFRα (CHO cells): 2.1 nM (Kd); PDGFRβ (CHO cells): 3.2 nM (Kd)

Form

Lyophilized powder

Purity

≥98%

Solubility

Warmed DMSO: 84 mg/mL (189.38 mM); Water: Insoluble; Ethanol: 7 mg/mL (15.78 mM)

Identity

Confirmed by NMR/HPLC/MS.

Applications

CP-868596 targets PDGFR, enabling investigations into its potential in disrupting cancer growth pathways.