PI3K inhibitor CH5132799, Purity ≥98%

Synonym: 1007207-67-1; CH-5132799; PI3K inhibitor

CAS Number: 1007207-67-1
Compound CID: 49784945

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

CH5132799, soluble in DMSO and insoluble in ethanol and water, is a potent compound that inhibits PI3 kinase activity. It targets PI3Kβ, PI3Kγ, C2α, C2β, mTOR, PI3Kα, PI3Kδ, and Vps34.

Molecular Weight

377.42

Molecular Formula

C₁₅H₁₉N₇O₃S

Targets

PI3Kβ: 0.12 μM; PI3Kγ: 1.6 μM; C2α: >10 μM; C2β: 5.3 μM; mTOR: 1.6 μM; PI3Kα: 14 nM; PI3Kδ: 0.50 μM; Vps34: >10 μM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 12 mg/mL (31.79 mM); Water: Insoluble; Ethanol: Insoluble

Identity

Confirmed by NMR/HPLC/MS.

Applications

CH5132799 can be used to study the inhibition of PI3K and mTOR signaling pathways in cancer cells.