PI3K inhibitor Pictilisib dimethanesulfonate, Purity ≥98%

Synonym: 957054-33-0; GDC-0941 dimethanesulfonate; GDC-0941 2 MeSO3H salt; PI3K inhibitor

CAS Number: 957054-33-0
Compound CID: 56972143

Product Size

50 mg; 100 mg; 500 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Pictilisib dimethanesulfonate is a potent compound that inhibits PI3 kinase activity. It targets Autophagy, DNA-PK, mTOR, p110α, p110α-E545K, p110α-H1047R, p110β, p110δ, and p110γ.

Molecular Weight

705.85

Molecular Formula

C₂₅H₃₅N₇O₉S₄

Targets

Autophagy; DNA-PK: 1.23 μM; mTOR: 0.58 μM; p110α: 3 nM; p110α-E545K: 3 nM; p110α-H1047R: 3 nM; p110β: 33 nM; p110δ: 3 nM; p110γ: 75 nM

Form

Lyophilized powder

Purity

≥98%

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

Pictilisib dimethanesulfonate can be used to inhibit PI3K signaling in cancer research.

Storage

Store at -20ºC.