PI3K inhibitor Pictilisib dimethanesulfonate, Purity ≥98%

Synonym: 957054-33-0; GDC-0941 dimethanesulfonate; GDC-0941 2 MeSO3H salt; PI3K inhibitor

CAS Number: 957054-33-0
Compound CID: 56972143

Product Size

50 mg; 100 mg; 500 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Pictilisib dimethanesulfonate is a potent compound that inhibits PI3 kinase activity. It targets Autophagy, DNA-PK, mTOR, p110α, p110α-E545K, p110α-H1047R, p110β, p110δ, and p110γ.

Molecular Weight

705.85

Molecular Formula

C₂₅H₃₅N₇O₉S₄

Targets

Autophagy; DNA-PK: 1.23 μM; mTOR: 0.58 μM; p110α: 3 nM; p110α-E545K: 3 nM; p110α-H1047R: 3 nM; p110β: 33 nM; p110δ: 3 nM; p110γ: 75 nM

Form

Lyophilized powder

Purity

≥98%

Identity

Confirmed by NMR/HPLC/MS.

Applications

Pictilisib dimethanesulfonate can be used to inhibit PI3K signaling in cancer research.