PI3K inhibitor SAR260301, Purity ≥98%

Synonym: 1260612-13-2; SAR 260301; SAR-260301; PI3K inhibitor

Product Size

5 mg; 10 mg; 50 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

SAR260301 is a potent compound that inhibits PI3 kinase activity. It targets DNA-PK, pAkt, PI3Kα, PI3Kβ, PI3Kδ, PI3Kγ, PI3KC2γ, and hsVps34.

Molecular Weight

354.4

Molecular Formula

C₁₉H₂₂N₄O₃

Targets

DNA-PK: 2000 nM; pAkt: 49 nM; PI3Kα: 1539 nM; PI3Kβ: 23 nM; PI3Kδ: 468 nM; PI3Kγ: 10000 nM; PI3KC2γ: 3812 nM; hsVps34: 183 nM

Form

Lyophilized powder

Purity

≥98%

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

SAR260301 is utilized to explore the inhibition of PI3K and its role in cellular signaling and cancer therapeutics.

Storage

Store at -20ºC.