PI3K inhibitor Tenalisib, Purity ≥98%

Synonym: 1639417-53-0; RP-6530; RP 6530; PI3K inhibitor

Product Size

2 mg; 5 mg; 25 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Tenalisib, soluble in DMSO and ethanol and insoluble in water, is a potent compound that inhibits PI3 kinase activity. It targets PI3Kδ and PI3Kγ.

Molecular Weight

415.43

Molecular Formula

C₂₃H₁₈FN₅O₂

Targets

PI3Kδ: 25 nM; PI3Kγ: 33 nM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 74 mg/mL (178.13 mM); Water: Insoluble; Ethanol: 74 mg/mL (178.13 mM)

Identity

Confirmed by NMR/HPLC/MS.

Stability

The product is stable for three years when stored at the recommended temperature in lyophilized powder.

Applications

Tenalisib is used to study the selective inhibition of PI3Kδ and its therapeutic potential in hematological malignancies and autoimmune diseases.

Storage

Store at -20ºC.