PI3K inhibitor Tenalisib, Purity ≥98%

Synonym: 1639417-53-0; RP-6530; RP 6530; PI3K inhibitor

Product Size

2 mg; 5 mg; 25 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

Tenalisib, soluble in DMSO and ethanol and insoluble in water, is a potent compound that inhibits PI3 kinase activity. It targets PI3Kδ and PI3Kγ.

Molecular Weight

415.43

Molecular Formula

C₂₃H₁₈FN₅O₂

Targets

PI3Kδ: 25 nM; PI3Kγ: 33 nM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 74 mg/mL (178.13 mM); Water: Insoluble; Ethanol: 74 mg/mL (178.13 mM)

Identity

Confirmed by NMR/HPLC/MS.

Applications

Tenalisib is used to study the selective inhibition of PI3Kδ and its therapeutic potential in hematological malignancies and autoimmune diseases.