PI3K inhibitor TG100-115, Purity ≥98%

Synonym: 677297-51-7; TG100115; PI3K inhibitor

CAS Number: 677297-51-7
Compound CID: 10427712

Product Size

5 mg; 10mg; 25 mg; 100 mg

Price

Datasheet

Datasheet

MSDS

MSDS

Properties

Description

TG100-115, soluble in DMSO and insoluble in ethanol and water, is a potent compound that inhibits PI3 kinase activity. It targets PI3Kα, PI3Kβ, PI3Kδ, and PI3Kγ.

Molecular Weight

346.3

Molecular Formula

C₁₈H₁₄N₆O₂

Targets

PI3Kα: 1.3 μM; PI3Kβ: 1.2 μM; PI3Kδ: 235 μM; PI3Kγ: 83 nM

Form

Lyophilized powder

Purity

≥98%

Solubility

DMSO: 8 mg/mL (23.09 mM); Water: Insoluble; Ethanol: Insoluble

Identity

Confirmed by NMR/HPLC/MS.

Applications

TG100-115 can be used to study the inhibition of PI3K and its downstream signaling in cancer and inflammatory responses.